Part I
General Part
Chapter I
Obtaining new drugs
Chapter II
Origin of Leads
Chapter III
Obtaining of compound libraries
Chapter IV
Pharmacokinetics
Chapter V
Pharmacodynamics
Chapter VI
Phase I metabolic reactions
Chapter VII
Phase II metabolic reactions
Chapter VIII
Toxic effects of metabolic bioactivation
Chapter IX
Receptors and drug activity
Chapter X
Enzymes
Chapter XI
Mechanism of action of drugs
Chapter XII
Stereochemistry and biological activity
Chapter XIII
Molecular Complications
Chapter XIV
Studies of structure-activity relationship (SAR)
Chapter XV
Change to the substituents in the lead
Chapter XVI
prodrugs
Chapter XVII
Pharmaceutical Forms
Chapter XVIII
biological membranes
Chapter XIX
Analysis of drugs and drug metabolites in complex matrices
Part II
Drugs acting on the central nervous system
Chapter XX
General anesthetics
Chapter XXI
Sedatives and hypnotics
Chapter XXII
Anticonvulsants
Chapter XXIII
opioid analgesics
Chapter XXIV
Antipsychotics
Chapter XXV
antiparkinson
Chapter XXVI
anxiolytics
Chapter XXVII
CNS stimulants (analeptic)
Chapter XXVIII
Antidepressants
Chapter XIX
Psychodysleptics (hallucinogens)
Chapter XXX
local anesthetics
Part III
Drugs acting on the autonomic nervous system and other drugs
Chapter XXXI
the cholinergic system Drugs
Chapter XXXII
Anticholinergic
Chapter XXXIII
adrenergic
Chapter XXXIV
Other antianginal and antihypertensive agents
Chapter XXXV
Cardiac glycosides and antiarrhythmic drugs
Chapter XXXVI
Antihistamines
Chapter XXXVII
Insight: Alzheimer's Disease
Chapter XXXIX
Diuretics